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Shp2 inhibitionSOS1PI3K/AKT signalingERK reactivationClinical trialCombination therapyCRCSotorasib resistanceTrametinibPMID: 39287412PMID: 34718292PMID: 35593017
EGFR feedback activation
MAPK reactivation
MEK dependency

Clinical Trials

Biomarkers

Mechanism

Literature

Protein Interactions

Resistance

Pathway Analysis

RMC-9805

92% evidence support

Research hypothesis — requires experimental validation

Refining evidence

312K pathways narrow to 24 candidates, then one strategy.

Filtering and prioritizing evidence…

Recommendation generated

From 41.7M evidence points to one therapeutic strategy.

312K pathways → 24 candidates → RMC-9805

Evidence considered

41.7M

data points

Pathways evaluated

312K

signaling pathways

Candidates considered

24

treatment strategies

Evidence support

92%

Literature · pathways · trials · resistance

KRAS G12D colorectal cancer✓ CompletedRMC-980592% evidence support

Research hypothesis — requires experimental validation · not a clinical recommendation

01

Funnel preserved

41.7M → 312K → 24 → 1

02

Evidence-linked

Every claim traces to sources

03

Actionable output

One strategy, with the why

Therapeutic Rationale

RMC-9805 is a selective KRAS G12D inhibitor with preclinical efficacy in colorectal cancer models. Strong on-target activity with a favorable safety profile.

KRAS G12D inhibitionTumor regressionHigh selectivity

Key Mechanism

KRAS G12DRAFMEKERK

RMC-9805 selectively targets KRAS G12D, preventing downstream MAPK pathway activation and tumor cell proliferation.

Evidence considered

41.7M

data points

Pathways evaluated

312K

signaling pathways

Candidates considered

24

treatment strategies

Evidence support

92%

literature · pathways · trials · resistance

Top Supporting Evidence

3 of 28 sources

Mutant-selective KRAS G12D inhibition in colorectal models

96%

Adaptive MAPK feedback following KRAS pathway blockade

92%

Biomarker stratification in KRAS G12D colorectal cancer

84%
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Our AI-driven analysis

41.7M

biomedical evidence points analyzed across publications, datasets, and clinical sources

312K

signaling pathways evaluated

24

treatment strategies considered

1

evidence-backed therapeutic strategy recommended